Tianeptine Free Acid Powder
Tianeptine free acid, a tricyclic compound, is a selective facilitator of 5-HT (serotonin) uptake in vitro and in vivo. In a study utilizing purified synaptosomes from rat brain, Tianeptine was reported to enhance serotonin uptake in selective brain regions. Has no affinity for a wide range of receptors, including 5-HT and dopamine (IC50 > 10 μM), and has no effect on noradrenalin or dopamine uptake. Antidepressant, analgesic and neuroprotective following systemic administration in vivo.
The benefits of taking a tianeptine free acid dose instead of a tianeptine sodium salt or sulfate dose can be profound. It provides the gentle sustained release of tianeptine sulfate, but without the hefty price tag. This allows for a more controlled dose and is the perfect form of tianeptine for those who are trying to reduce the amount of tianeptine they intake daily. For those who want a more concentrated dose of tianeptine, you can convert tianeptine free acid into sodium salt with relative ease.
Tianeptine Free Acid Basic Info
Product name: Tianeptine acid
Appearance White powder
Solubility DMSO: ≥20 mg/mL
Assay ≥99% (HPLC)