Tianeptine Free Acid

Tianeptine Free Acid PowderTianeptine Free Acid.jpg

Tianeptine free acid, a tricyclic compound, is a selective facilitator of 5-HT (serotonin) uptake in vitro and in vivo.  In a study utilizing purified synaptosomes from rat brain, Tianeptine was reported to enhance serotonin uptake in selective brain regions.  Has no affinity for a wide range of receptors, including 5-HT and dopamine (IC50 > 10 μM), and has no effect on noradrenalin or dopamine uptake. Antidepressant, analgesic and neuroprotective following systemic administration in vivo.

The benefits of taking a tianeptine free acid dose instead of a tianeptine sodium salt or sulfate dose can be profound. It provides the gentle sustained release of tianeptine sulfate, but without the hefty price tag. This allows for a more controlled dose and is the perfect form of tianeptine for those who are trying to reduce the amount of tianeptine they intake daily. For those who want a more concentrated dose of tianeptine, you can convert tianeptine free acid into sodium salt with relative ease.

Tianeptine Free Acid Basic Info 

Product name: Tianeptine acid
CAS:    66981-73-5
MF:    C21H25ClN2O4S
MW:    436.95
Appearance    White powder
Solubility    DMSO: ≥20 mg/mL
Assay    ≥99% (HPLC)

 

Author: chemicals

Here is chemical sourse

Leave a Reply

Fill in your details below or click an icon to log in:

WordPress.com Logo

You are commenting using your WordPress.com account. Log Out / Change )

Twitter picture

You are commenting using your Twitter account. Log Out / Change )

Facebook photo

You are commenting using your Facebook account. Log Out / Change )

Google+ photo

You are commenting using your Google+ account. Log Out / Change )

Connecting to %s